SCHEMBL29656385

SCHEMBL29656385

COC(=O)c1cnc2[nH]ccc2c1N

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TTBK1 Q5TCY1 1/20 0.48
TTBK2 Q6IQ55 1/20 0.48
AXL P30530 5/20 0.46
NUDT1 P36639 1/20 0.46
MAP2K1 Q02750 1/20 0.46
TSHR P16473 1/20 0.44
JAK1 P23458 9/20 0.43
JAK3 P52333 9/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
JAK2 O60674 5/20 0.43
CDK8 P49336 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28798529 1.00 TTBK1 (0.48) TTBK1TTBK2AXLNUDT1MAP2K1
SCHEMBL20990227 0.86 NUDT1 (0.65) NUDT1JAK1JAK3
SCHEMBL2632955 0.83 NUDT1 (0.50) TTBK1TTBK2AXLNUDT1MAP2K1
SCHEMBL31403755 0.83 NUDT1 (0.50) TTBK1TTBK2AXLNUDT1MAP2K1
SCHEMBL12876743 0.83 JAK2 (0.53) NUDT1JAK1JAK3JAK2
SCHEMBL2359607 0.83 HAVCR2 (0.48) AXLNUDT1MAP2K1JAK1JAK3
SCHEMBL25280494 0.82 AXL (0.46) TTBK1TTBK2AXLNUDT1MAP2K1
SCHEMBL21632535 0.82 JAK3 (0.46) TTBK1TTBK2AXLNUDT1MAP2K1
SCHEMBL31403683 0.82 JAK3 (0.46) TTBK1TTBK2AXLNUDT1MAP2K1
SCHEMBL30985188 0.82 AXL (0.55) TTBK1TTBK2AXLNUDT1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114539245-A Pyrimidine-fused ring derivative-containing regulator, and preparation method and application thereof 上海翰森生物医药科技有限公司 2022-05-27 CN disclosed