SCHEMBL2529112

SCHEMBL2529112

FC(F)(F)c1ccccc1-c1ccccc1-c1cccnc1-c1ccccc1-c1ccccc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 2/20 0.48
CTSL P07711 1/20 0.48
CTSS P25774 1/20 0.48
PTPN13 Q12923 1/20 0.48
CYP3A4 P08684 7/20 0.44
CYP1A2 P05177 6/20 0.44
CYP2C19 P33261 5/20 0.44
CYP2D6 P10635 4/20 0.44
TDP1 Q9NUW8 3/20 0.44
MEN1 O00255 1/20 0.44
THRB P10828 1/20 0.44
BLM P54132 1/20 0.44
KMT2A Q03164 1/20 0.44
PDK2 Q15119 1/20 0.44
HSD11B1 P28845 1/20 0.43
ALOX15 P16050 3/20 0.43
HSD17B10 Q99714 3/20 0.43
MAPK1 P28482 2/20 0.43
ALDH1A1 P00352 2/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12854133 1.00 PTPRC (0.48) PTPRCCTSLCTSSPTPN13CYP3A4
SCHEMBL27924774 0.94 CYP3A4 (0.46) PTPRCCTSLCTSSPTPN13CYP3A4
SCHEMBL14124513 0.91 HSD11B1 (0.44) PTPRCCTSLCTSSPTPN13CYP3A4
SCHEMBL12854126 0.85 ALDH1A1 (0.48) CYP3A4CYP1A2CYP2C19CYP2D6TDP1
SCHEMBL11910213 0.82 PTPRC (0.67) PTPRCCTSLCTSSPTPN13CYP3A4
SCHEMBL22929973 0.82 PTPRC (0.67) PTPRCCTSLCTSSPTPN13CYP3A4
SCHEMBL14935529 0.82 PTPRC (0.67) PTPRCCTSLCTSSPTPN13CYP3A4
SCHEMBL28420415 0.82 PTPRC (0.67) PTPRCCTSLCTSSPTPN13CYP3A4
SCHEMBL28273066 0.81 PTPRC (0.44) PTPRCCTSLCTSSPTPN13CYP3A4
SCHEMBL8022901 0.79 HSD11B1 (0.54) CYP3A4CYP1A2CYP2C19CYP2D6TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2375904-A1 BIARYL CARBOXAMIDES Merck Sharp & Dohme Corp. (US) 2011-10-19 EP claimed