SCHEMBL25328822

SCHEMBL25328822

COc1ccc(-c2csc(NN)n2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.70
MAPT P10636 8/20 0.68
RAB9A P51151 8/20 0.68
MEN1 O00255 8/20 0.68
KMT2A Q03164 8/20 0.68
SMN1; SMN2 Q16637 7/20 0.68
NPC1 O15118 6/20 0.68
GAA P10253 4/20 0.68
ALDH1A1 P00352 4/20 0.66
POLB P06746 1/20 0.66
NFKB1 P19838 4/20 0.65
NFKB2 Q00653 4/20 0.65
RELA Q04206 4/20 0.65
ALOX5 P09917 3/20 0.65
MCL1 Q07820 1/20 0.65
VCP P55072 1/20 0.62
GFER P55789 1/20 0.61
RECQL P46063 1/20 0.61
MAPK1 P28482 2/20 0.60
TUBB4A P04350 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24590341 0.85 PTGS2 (0.72) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL12297852 0.83 PTGS2 (1.00) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL7537503 0.83 PTGS2 (1.00) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL30118253 0.82 NPC1 (0.68) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL28911472 0.82 NPC1 (0.68) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL28030442 0.81 MAPT (0.67) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL24590327 0.81 RAB9A (0.68) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL24590324 0.81 PTGS2 (0.67) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL24590148 0.81 PTGS2 (0.67) PTGS2MAPTRAB9AMEN1KMT2A
SCHEMBL3595657 0.81 PTGS2 (0.66) PTGS2MAPTRAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023141262-A1 BAX ACTIVATORS AND USE THEREOF IPSEN PHARMA S.A.S. (FR) 2023-07-27 WO disclosed
WO-2023141262-A1 BAX ACTIVATORS AND USE THEREOF IPSEN PHARMA S.A.S. (FR) 2023-07-27 WO disclosed
CN-113880786-B Synthesis method and anti-oxidation application of camphene aldehyde thiazole hydrazone derivative 江西农业大学 2023-03-03 CN disclosed
CN-115448915-A SIRT5 inhibitor and preparation method and application thereof 广西师范大学 2022-12-09 CN disclosed