SCHEMBL25337498

SCHEMBL25337498

CC(C)CCN(C(=O)O)[C@@H]1CCc2cc(OCc3ccccc3)c(Br)c(F)c2C1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.35
HTR2A P28223 2/20 0.35
HTR2C P28335 1/20 0.35
TRPM8 Q7Z2W7 4/20 0.34
S1PR5 Q9H228 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
CACNA1B Q00975 1/20 0.33
UBE2M P61081 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33
MMP2 P08253 1/20 0.33
MMP13 P45452 1/20 0.33
AGTR2 P50052 1/20 0.33
GLRA1 P23415 1/20 0.33
TAOK1 Q7L7X3 1/20 0.33
TAOK3 Q9H2K8 1/20 0.33
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29132505 0.93 HTR2A (0.38) MC4RHTR2A
SCHEMBL25339129 0.90 MC4R (0.37) MC4RTRPM8S1PR5MEN1NPC1
SCHEMBL25340719 0.84 GHSR (0.34) MC4RMEN1NPC1RAB9AKMT2A
SCHEMBL29132480 0.82 HTR2A (0.38) MC4RHTR2ATRPM8
SCHEMBL29626276 0.82 HTR2A (0.38) MC4RHTR2ATRPM8
SCHEMBL25340552 0.81 PTPN2 (0.49)
SCHEMBL25339199 0.78 PTPN2 (0.43) HTR2AHTR2CMEN1NPC1RAB9A
SCHEMBL29132471 0.78 RORC (0.35) HTR2A
SCHEMBL29626362 0.77 HTR2A (0.35) HTR2AMEN1NPC1RAB9AKMT2A
SCHEMBL25338586 0.76 ITGB3 (0.43) HTR2AHTR2CS1PR5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4211122-A1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Calico Life Sciences LLC (US) 2023-07-19 EP disclosed