SCHEMBL25352121

SCHEMBL25352121

CS(=O)(=O)Nc1cc(Cl)cc(NC(=O)c2cccc(-n3ccc(C#N)n3)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HTT P42858 3/20 0.41
MAPT P10636 3/20 0.41
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
HPGD P15428 2/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
DHX9 Q08211 1/20 0.40
EGFR P00533 2/20 0.39
FGFR1 P11362 2/20 0.39
KDR P35968 2/20 0.39
RIPK1 Q13546 1/20 0.39
USP36 Q9P275 1/20 0.39
EPHX2 P34913 1/20 0.39
MAPK10 P53779 3/20 0.39
GPR142 Q7Z601 2/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30535297 1.00 MEN1 (0.41) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL25350503 0.85 HTT (0.43) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL30535005 0.85 HTT (0.43) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL25430854 0.83 DHX9 (0.42) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL30535450 0.83 DHX9 (0.42) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL25351911 0.82 KAT6A (0.51) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL30535596 0.82 KAT6A (0.51) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL31057061 0.75 TNIK (0.50) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL25430853 0.75 TNIK (0.50) MEN1KMT2AHTTMAPTALDH1A1
SCHEMBL31561256 0.74 MEN1 (0.45) MEN1KMT2AHTTMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154519-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed
WO-2023154519-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed