SCHEMBL30535005

SCHEMBL30535005

CS(=O)(=O)Nc1cc(Cl)cc(NC(=O)c2cccc(-n3ccc(CO)n3)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.43
MEN1 O00255 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 2/20 0.42
KDM4E B2RXH2 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
DHX9 Q08211 1/20 0.41
KAT6A Q92794 1/20 0.40
EGFR P00533 2/20 0.40
FGFR1 P11362 2/20 0.40
KDR P35968 2/20 0.40
USP36 Q9P275 1/20 0.40
MAPK10 P53779 4/20 0.40
GPR142 Q7Z601 2/20 0.40
KCNK3 O14649 2/20 0.39
KCNK9 Q9NPC2 1/20 0.39
MAPK8 P45983 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25350503 1.00 HTT (0.43) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL31561256 0.89 MEN1 (0.45) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL30535450 0.85 DHX9 (0.42) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL25352121 0.85 MEN1 (0.41) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL25430854 0.85 DHX9 (0.42) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL30535297 0.85 MEN1 (0.41) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL25351911 0.83 KAT6A (0.51) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL30535596 0.83 KAT6A (0.51) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL25353685 0.73 KAT6A (0.51) HTTMEN1ALDH1A1KMT2AMAPT
SCHEMBL30535678 0.73 KAT6A (0.51) HTTMEN1ALDH1A1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250145597-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. 2025-05-08 US disclosed
CN-119923385-A Inhibitors of RNA helicase DHX9 and uses thereof 埃克森特治疗公司 2025-05-02 CN disclosed
WO-2025080900-A1 INHIBITORS OF THE RNA HELICASE DHX9 FOR USE IN THE TREATMENT OF DNA DAMAGE REPAIR DEFICIENT, HOMOLOGOUS RECOMBINATION DEFICIENT, AND CANCERS HAVING A BRCA LOSS OF FUNCTION MUTATION ACCENT THERAPEUTICS, INC. (US) 2025-04-17 WO disclosed
US-12233065-B2 Inhibitors of RNA helicase DHX9 and uses thereof ACCENT THERAPEUTICS, INC. (US) 2025-02-25 US disclosed
EP-4479138-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF Accent Therapeutics, Inc. (US) 2024-12-25 EP disclosed
US-12162867-B2 Inhibitors of RNA helicase DHX9 and uses thereof ACCENT THERAPEUTICS, INC. (US) 2024-12-10 US disclosed
US-20240316047-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. 2024-09-26 US disclosed
US-20240279210-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. 2024-08-22 US disclosed
WO-2023154519-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. (US) 2023-08-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240316047-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF DHX29, DHX9, DDX39B HTT 1061/4885MEN1 3318/4885ALDH1A1 1705/4885
US-20240279210-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF DHX29, DHX9, DDX39B HTT 1177/4885MEN1 3191/4885ALDH1A1 1333/4885
US-12233065-B2 Inhibitors of RNA helicase DHX9 and uses thereof DHX29, DHX9, DDX39B HTT 1061/4885MEN1 3318/4885ALDH1A1 1705/4885
US-12162867-B2 Inhibitors of RNA helicase DHX9 and uses thereof DHX29, DHX9, DDX39B HTT 1177/4885MEN1 3191/4885ALDH1A1 1333/4885
US-20250145597-A1 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF DHX9, DHX29, DDX39B HTT 1031/4885MEN1 3047/4885ALDH1A1 1127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.