SCHEMBL25404705

SCHEMBL25404705

COC(=O)c1cc(F)c(N)c(NCC2CCO2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
PTGER4 P35408 2/20 0.39
HPGD P15428 5/20 0.38
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 1/20 0.37
HCAR3 P49019 1/20 0.36
TDO2 P48775 1/20 0.36
BACE1 P56817 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 1/20 0.35
GAA P10253 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25279173 1.00 KMT2A (0.40) KMT2APTGER4HPGDALDH1A1KDM4E
SCHEMBL31463429 1.00 KMT2A (0.40) KMT2APTGER4HPGDALDH1A1KDM4E
SCHEMBL30393343 0.90 KMT2A (0.43) KMT2AHPGDALDH1A1KDM4EHCAR3
SCHEMBL28754429 0.90 PTGER4 (0.47) KMT2APTGER4HPGDALDH1A1KDM4E
SCHEMBL29640515 0.90 PTGER4 (0.47) KMT2APTGER4HPGDALDH1A1KDM4E
SCHEMBL23286839 0.90 PTGER4 (0.47) KMT2APTGER4HPGDALDH1A1KDM4E
SCHEMBL24901946 0.88 PTGER4 (0.43) KMT2APTGER4HPGDALDH1A1KDM4E
SCHEMBL30232663 0.88 PTGER4 (0.43) KMT2APTGER4HPGDALDH1A1KDM4E
SCHEMBL28754443 0.86 HCAR3 (0.46) KMT2AHPGDALDH1A1KDM4EHCAR3
SCHEMBL28754455 0.86 HCAR3 (0.46) KMT2AHPGDALDH1A1KDM4EHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023222124-A1 5,6-DIHYDRO-1,2,4-TRIAZINE COMPOUND AND PHARMACEUTICAL USE THEREOF AS GLP-1 RECEPTOR AGONIST 中国科学院上海药物研究所 2023-11-23 WO disclosed
WO-2023169436-A1 BENZO BICYCLIC COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF 广州市联瑞制药有限公司 2023-09-14 WO disclosed