SCHEMBL254093

SCHEMBL254093

CC(C)Cc1ccc(C(=O)c2ccc(C(N)=O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.56
ALOX5 P09917 2/20 0.50
PTGS1 P23219 4/20 0.49
PTGS2 P35354 4/20 0.49
CXCR1 P25024 3/20 0.49
CXCR2 P25025 3/20 0.49
LMNA P02545 3/20 0.49
CYP2C9 P11712 2/20 0.49
AKR1C3 P42330 2/20 0.49
ALB P02768 1/20 0.49
ESR1 P03372 1/20 0.49
RARB P10826 1/20 0.49
ADRB3 P13945 1/20 0.49
NFKB1 P19838 1/20 0.49
HTR2A P28223 1/20 0.49
NR1I3 Q14994 1/20 0.49
SLC22A6 Q4U2R8 1/20 0.49
CXCL8 P10145 1/20 0.49
TSHR P16473 1/20 0.49
AKR1C2 P52895 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL105246 0.94 EPHX1 (0.61) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL21064585 0.90 PTGS1 (0.57) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL13718987 0.89 EPHX1 (0.56) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL10580349 0.85 EPHX1 (0.51) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL5018743 0.83 PTGS1 (0.55) ALOX5PTGS1PTGS2CXCR1CXCR2
SCHEMBL25693884 0.83 LMNA (0.61) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL24827555 0.81 TRPA1 (0.50) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL8745472 0.81 TAAR1 (0.59) PLA2G10PLA2G2A
SCHEMBL6764390 0.81 TAAR1 (0.59) PLA2G10PLA2G2A
SCHEMBL9392575 0.81 TAAR1 (0.59) PLA2G10PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2459565-B1 SAXITOXIN DERIVATIVES, METHODS AND COMPOSITIONS FOR STUDYING, IMAGING, AND TREATING PAIN UNIV LELAND STANFORD JUNIOR (US) 2018-05-02 EP disclosed
WO-2010129864-A9 METHODS AND COMPOSITIONS FOR STUDYING, IMAGING, AND TREATING PAIN THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2012-03-08 WO disclosed
WO-2010129864-A2 METHODS AND COMPOSITIONS FOR STUDYING, IMAGING, AND TREATING PAIN THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2010-11-11 WO disclosed