SCHEMBL25439485

SCHEMBL25439485

COC(=O)c1cnc(C(=O)c2ccc(F)cc2)n1COCC[Si](C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 3/20 0.38
NPC1 O15118 6/20 0.37
KDM5A P29375 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
PTGS2 P35354 1/20 0.35
MAPT P10636 5/20 0.35
RAB9A P51151 4/20 0.35
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
HTT P42858 3/20 0.35
LMNA P02545 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HPGD P15428 2/20 0.35
S1PR4 O95977 1/20 0.35
S1PR1 P21453 1/20 0.35
PPARG P37231 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
NCOA2 Q15596 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27398571 0.89 NPC1 (0.39) GABRA5NPC1PTGS2MAPTRAB9A
SCHEMBL30889520 0.77 MAPT (0.37) NPC1MAPTRAB9ASMN1; SMN2DGAT1
SCHEMBL22112683 0.70 THRB (0.38) NPC1MAPTRAB9ASMN1; SMN2LMNA
SCHEMBL25258361 0.70 F11 (0.39) NPC1MAPTRAB9AALDH1A1SMN1; SMN2
SCHEMBL31629099 0.70 GRIN2B (0.38) MAPTRAB9AALDH1A1MEN1MAPK1
SCHEMBL3076793 0.69 NPC1 (0.42) NPC1MAPTDGAT1
SCHEMBL30903072 0.69 NPC1 (0.36) NPC1MAPTRAB9AALDH1A1SMN1; SMN2
SCHEMBL30867579 0.69 DGAT1 (0.39) GABRA5NPC1MAPTRAB9AALDH1A1
SCHEMBL25911833 0.69 F2RL1 (0.36) NPC1KDM5AKDM5BMAPTALDH1A1
SCHEMBL30903056 0.68 NPC1 (0.35) NPC1MAPTRAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118613483-A Plasma kallikrein inhibitors 默沙东有限责任公司 2024-09-06 CN disclosed
WO-2023146809-A9 PLASMA KALLIKREIN INHIBITORS MERCK SHARP & DOHME LLC (US) 2024-03-14 WO disclosed
WO-2023146809-A1 PLASMA KALLIKREIN INHIBITORS MERCK SHARP & DOHME LLC (US) 2023-08-03 WO disclosed