SCHEMBL25453080

SCHEMBL25453080

CN(c1ccccc1)c1ccc(N)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.46
EGFR P00533 3/20 0.45
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CSF1R P07333 2/20 0.39
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
PDE4A P27815 1/20 0.35
TP53 P04637 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
HDAC1 Q13547 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30639141 0.90 ALDH1A1 (0.43) DHFREGFRALDH1A1CYP3A4TDP1
SCHEMBL6754283 0.80 L3MBTL1 (0.46) ALDH1A1KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL22453529 0.78 ALDH1A1 (0.33) DHFRALDH1A1CYP3A4TDP1TP53
SCHEMBL30488787 0.78 GBA1 (0.50) DHFREGFRALDH1A1KDM4EMAPT
SCHEMBL25301327 0.78 GBA1 (0.50) DHFREGFRALDH1A1KDM4EMAPT
SCHEMBL28504853 0.77 HDAC6 (0.49) DHFREGFRALDH1A1CYP3A4TDP1
SCHEMBL29618352 0.76 ALDH1A1 (0.42) ALDH1A1CYP3A4TDP1KDM4ETP53
SCHEMBL142308 0.76 ALDH1A1 (0.42) ALDH1A1CYP3A4TDP1KDM4ETP53
SCHEMBL12016060 0.75 KDM4C (0.44) DHFREGFRTDP1KDM4EMAPT
SCHEMBL5206210 0.74 CYP2D6 (0.44) DHFREGFRALDH1A1CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2671575-A1 Ras inhibitors Universität Regensburg (DE) 2013-12-11 EP claimed
WO-2023081800-A1 ALPHA-2A ADRENERGIC RECEPTOR MODULATORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-05-11 WO disclosed
EP-2671575-A1 Ras inhibitors Universität Regensburg (DE) 2013-12-11 EP disclosed