SCHEMBL254535

SCHEMBL254535

C[C@@H](O)[C@H](NS(=O)(=O)c1ccc(-c2ccc(N)cc2)cc1)C(=O)NO

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 9/20 0.65
MMP9 P14780 9/20 0.65
MMP13 P45452 9/20 0.65
MMP7 P09237 8/20 0.65
MMP2 P08253 8/20 0.65
MMP3 P08254 7/20 0.65
ADAM17 P78536 2/20 0.59
MMP14 P50281 2/20 0.59
ADAM10 O14672 1/20 0.59
MMP8 P22894 1/20 0.59
ALDH1A1 P00352 1/20 0.51
SLC1A3 P43003 1/20 0.51
SLC1A2 P43004 1/20 0.51
SLC1A1 P43005 1/20 0.51
ADAMTS4 O75173 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL405125 0.88 MMP9 (0.66) MMP1MMP9MMP13MMP7MMP2
SCHEMBL4915104 0.88 MMP9 (0.66) MMP1MMP9MMP13MMP7MMP2
SCHEMBL15228196 0.86 MMP9 (0.59) MMP1MMP9MMP13MMP7MMP2
SCHEMBL174865 0.86 MMP9 (0.59) MMP1MMP9MMP13MMP7MMP2
SCHEMBL255126 0.85 MMP2 (0.67) MMP1MMP9MMP13MMP7MMP2
SCHEMBL4916984 0.83 MMP9 (0.60) MMP1MMP9MMP13MMP7MMP2
SCHEMBL14025839 0.83 MMP9 (0.60) MMP1MMP9MMP13MMP7MMP2
SCHEMBL4431428 0.79 MMP2 (1.00) MMP1MMP9MMP13MMP7MMP2
SCHEMBL3618803 0.79 MMP2 (1.00) MMP1MMP9MMP13MMP7MMP2
SCHEMBL7082523 0.78 MMP2 (1.00) MMP1MMP9MMP13MMP7MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed