SCHEMBL255126

SCHEMBL255126

COC(=O)[C@@H](NS(=O)(=O)c1ccc(-c2ccc(N)cc2)cc1)[C@@H](C)O

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 12/20 0.67
MMP9 P14780 10/20 0.67
MMP3 P08254 10/20 0.67
MMP13 P45452 10/20 0.67
MMP1 P03956 9/20 0.67
MMP7 P09237 9/20 0.67
MMP8 P22894 1/20 0.53
SLC1A3 P43003 1/20 0.52
SLC1A2 P43004 1/20 0.52
SLC1A1 P43005 1/20 0.52
ADAMTS4 O75173 4/20 0.51
MMP14 P50281 1/20 0.49
ALDH1A1 P00352 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1110930 0.92 MMP2 (0.75) MMP2MMP9MMP3MMP13MMP1
SCHEMBL1110927 0.92 MMP2 (0.75) MMP2MMP9MMP3MMP13MMP1
SCHEMBL3607214 0.92 MMP2 (0.75) MMP2MMP9MMP3MMP13MMP1
SCHEMBL15235737 0.86 MMP9 (0.50) MMP2MMP9MMP3MMP13MMP1
SCHEMBL254535 0.85 MMP1 (0.65) MMP2MMP9MMP3MMP13MMP1
SCHEMBL3608987 0.85 MMP2 (0.58) MMP2MMP9MMP3MMP13MMP1
SCHEMBL156173 0.81 MMP9 (0.47) MMP2MMP9MMP3MMP13MMP1
SCHEMBL3618803 0.80 MMP2 (1.00) MMP2MMP9MMP3MMP13MMP1
SCHEMBL4431428 0.80 MMP2 (1.00) MMP2MMP9MMP3MMP13MMP1
SCHEMBL14045736 0.80 ADAMTS4 (0.64) MMP2MMP9MMP3MMP13MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed