Racemoramide

Racemoramide

SCHEMBL25463

C[C@H](CN1CCOCC1)C(C(=O)N1CCCC1)(c1ccccc1)c1ccccc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.51
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
NPC1 O15118 2/20 0.50
MEN1 O00255 8/20 0.48
KMT2A Q03164 8/20 0.48
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ATM Q13315 2/20 0.44
HTT P42858 2/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
HIF1A Q16665 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Levomoramide SCHEMBL907811 1.00 SMN1; SMN2 (0.51) SMN1; SMN2ALDH1A1LMNANPC1MEN1
Racemoramide SCHEMBL548434 1.00 SMN1; SMN2 (0.51) SMN1; SMN2ALDH1A1LMNANPC1MEN1
Racemoramide SCHEMBL7474188 0.98 SMN1; SMN2 (0.49) SMN1; SMN2ALDH1A1LMNANPC1MEN1
Racemoramide SCHEMBL548433 0.94 SMN1; SMN2 (0.46) SMN1; SMN2ALDH1A1LMNANPC1MEN1
SCHEMBL9917087 0.93 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1LMNANPC1MEN1
SCHEMBL9917086 0.88 KDM4E (0.46) SMN1; SMN2ALDH1A1LMNANPC1MEN1
SCHEMBL22313199 0.88 L3MBTL1 (0.52) SMN1; SMN2ALDH1A1LMNANPC1MEN1
Racemoramide SCHEMBL8741247 0.86 ADRA2B (0.44) SMN1; SMN2ALDH1A1LMNANPC1MEN1
SCHEMBL17028079 0.86 ALDH1A1 (0.56) SMN1; SMN2ALDH1A1LMNANPC1MEN1
SCHEMBL22313196 0.85 SMN1; SMN2 (0.46) SMN1; SMN2ALDH1A1LMNANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10741 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
EP-4714444-A1 PREPARATION FOR AND USE OF CANNABIDIOL DERIVATIVE DRUGS Changchun Institute Of Applied Chemistry Chinese Academy Of Sciences (CN) 2026-03-25 EP claimed
EP-4100010-B1 NITROXIDE COMPOUNDS FOR USE IN THE TREATMENT OF OPIOID-INDUCED RESPIRATORY DEPRESSION (OIRD) UNIV CASE WESTERN RESERVE (US) 2026-01-07 EP claimed
US-20250326778-A1 PYRAZOLE COMPOUNDS AND METHOD FOR MAKING AND USING THE COMPOUNDS RIGEL PHARMACEUTICALS, INC. (US) 2025-10-23 US claimed
US-20250319074-A1 TREATMENT AND MANAGEMENT OF AUGMENTATION IN RESTLESS LEGS SYNDROME UNIV EAST CAROLINA (US) 2025-10-16 US claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-12383743-B2 Treatment of addiction and dependency TACA JR ARTURO C (US) 2025-08-12 US claimed
US-20250228771-A1 ALKALINE INTRAORAL PRODUCTS EMPLICURE AB (publ) (SE) 2025-07-17 US claimed
EP-4581017-A1 NEW N-HETEROARYLBENZAMIDES DERIVATIVES AS FLT3 INHIBITORS Biodol Therapeutics (FR) 2025-07-09 EP claimed
EP-0415693-A1 Composition and method for selective enhancement of opiate activity and reduction of opiate tolerance and dependence ARIZONA TECHNOLOGY DEVELOPMENT CORPORATION (US) 1991-03-06 EP claimed
EP-0377518-A2 Sustained release pharmaceutical composition F.H. FAULDING & CO. LIMITED (AU) 1990-07-11 EP claimed
EP-0174342-B1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1989-12-20 EP claimed
US-4879298-A ADMINISTERING FORSKOLINE TO POTENTIATE ANALGESIC EFFECTS OF NARCOTICS ROUSSEL UCLAF (FR) 1989-11-07 US claimed
EP-0287469-A1 Mixture containing as the active principles a central analgesic and forskolin ROUSSEL-UCLAF (FR) 1988-10-19 EP claimed
US-4760070-A Administering central analgesic and sufficient adenine ROUSSEL UCLAF (FR) 1988-07-26 US claimed
EP-0108017-B1 MIXTURE COMPRISING A CENTRAL ANALGESIC AND VITAMIN B12, OR ONE OF ITS ANALOGS, AS ACTIVE PRINCIPLES ROUSSEL-UCLAF (FR) 1986-12-10 EP claimed
US-4522816-A VITAMIN B12 OR DERIVATIVE ADDED TO POTENTIALIZE CENTRAL ANALGESIC WITH REDUCED TOXICITY ROUSSEL UCLAF (FR) 1985-06-11 US claimed
US-4126684-A 4-AMINO-3-P-HALOPHENYLBUTYRIC ACIDS AND THEIR DERIVATIVES USED IN THE CONTROL OF NARCOTIC ABUSE CIBA-GEIGY CORPORATION (US) 1978-11-21 US claimed
US-4053604-A 3-HYDROXY-3-ISOPROPYL-2,3,4,4A,8,9,13B,14-OCTAHYDRO-1H -BENZO(6,7)CYCLOPENTA(1,2,3-DE)PYRIDO(2,1-A)ISOQUINOLIN-3-OL AYERST, MCKENNA & HARRISON LIMITED (CA) 1977-10-11 US claimed