SCHEMBL25466554

SCHEMBL25466554

COC(C)(C)c1ncc2ccc(=O)[nH]c2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32
HTR2A P28223 1/20 0.32
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CDK7 P50613 1/20 0.30
CCNH P51946 1/20 0.30
MNAT1 P51948 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
GLA P06280 1/20 0.30
PMP22 Q01453 1/20 0.30
HSD17B10 Q99714 1/20 0.30
HCAR1 Q9BXC0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21455110 0.84 MAPK8 (0.39) MAPK8MAPK9MAPK10PDE3BPDE3A
SCHEMBL29828263 0.78 MAPK8 (0.36) MAPK8MAPK9MAPK10PDE3BPDE3A
SCHEMBL4129449 0.74 DYRK1A (0.41) MAPK8MAPK9MAPK10PDE3BPDE3A
SCHEMBL29641025 0.73 CA12 (0.36) MAPK8MAPK9MAPK10PDE3BPDE3A
SCHEMBL23264212 0.72 NUDT1 (0.31)
SCHEMBL3334033 0.72 PDE3B (0.44) MAPK8MAPK9MAPK10PDE3BPDE3A
SCHEMBL19019072 0.71 PDE3B (0.38) MAPK8MAPK9MAPK10PDE3BPDE3A
SCHEMBL16416249 0.69 MAPK8 (0.48) MAPK8MAPK9MAPK10PDE3BPDE3A
SCHEMBL29837916 0.69 HTR1A (0.44) MAPK8MAPK9MAPK10PDE3BPDE3A
SCHEMBL1983844 0.68 ALDH1A1 (0.43) MAPK8MAPK9MAPK10PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023083297-A1 SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2023-05-19 WO disclosed