SCHEMBL25470355

SCHEMBL25470355

CC(C)(C)OC(=O)NCc1ccccc1-c1cc(N)c(F)cc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 3/20 0.52
KDM4A O75164 1/20 0.43
ALOX5AP P20292 1/20 0.41
FEN1 P39748 1/20 0.41
HDAC1 Q13547 1/20 0.41
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
MALT1 Q9UDY8 1/20 0.39
RIPK1 Q13546 1/20 0.39
IDO1 P14902 1/20 0.39
PDK2 Q15119 1/20 0.38
NQO2 P16083 1/20 0.38
BRD9 Q9H8M2 1/20 0.38
BAZ2B Q9UIF8 1/20 0.38
BAZ2A Q9UIF9 1/20 0.38
GRM2 Q14416 1/20 0.38
BRD4 O60885 1/20 0.38
RPS6KA1 Q15418 1/20 0.38
PTPN1 P18031 1/20 0.37
HDAC10 Q969S8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25470479 0.88 KCNA5 (0.50) KCNA5KDM4AALOX5APFEN1HDAC1
SCHEMBL25471591 0.85 AAK1 (0.45) KCNA5KDM4AALOX5APFEN1HDAC1
SCHEMBL29467997 0.82 KDM4A (0.41) KCNA5KDM4AHDAC1CTSSCTSK
SCHEMBL25471532 0.82 KCNA5 (0.53) KCNA5KDM4AHDAC1MALT1NQO2
SCHEMBL31296532 0.80 SCN9A (0.50) ALOX5APFEN1MALT1IDO1PDK2
SCHEMBL25470614 0.80 SCN9A (0.50) ALOX5APFEN1MALT1IDO1PDK2
SCHEMBL2002789 0.80 KDM4A (0.41) KCNA5KDM4AHDAC1CTSSCTSK
SCHEMBL25470761 0.79 MALT1 (0.45) KCNA5KDM4AALOX5APFEN1MALT1
SCHEMBL8254926 0.79 KCNA5 (0.61) KCNA5KDM4AHDAC1MALT1IDO1
SCHEMBL4590703 0.78 RIPK1 (0.60) KCNA5KDM4ACTSSCTSKRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078127-A1 MACROCYCLIC SULFONAMIDE COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 中国药科大学 2023-05-11 WO disclosed