SCHEMBL254900

SCHEMBL254900

C[C@@](O)(C(F)F)[C@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(=O)NO

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 5/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19262730 0.89
SCHEMBL19520703 0.89 ADAMTS5 (0.47) ANPEPNPC1RAB9A
SCHEMBL19534376 0.89 ADAMTS5 (0.47) ANPEPNPC1RAB9A
SCHEMBL19520702 0.89 ADAMTS5 (0.47) ANPEPNPC1RAB9A
SCHEMBL21082092 0.88 ANPEP (0.40) ANPEP
SCHEMBL21046331 0.87
SCHEMBL15235778 0.87
SCHEMBL15227416 0.87
SCHEMBL255220 0.87 NPC1 (0.41) NPC1RAB9A
SCHEMBL21046243 0.86 ANPEP (0.38) ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed