SCHEMBL2551595

SCHEMBL2551595

O=S(=O)(c1ccc(CN2CCNCC2)cc1)N1CCCC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.58
MAPT P10636 1/20 0.58
USP2 O75604 1/20 0.56
CXCR4 P61073 4/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
CHRM2 P08172 1/20 0.55
CHRM1 P11229 1/20 0.55
ADRA2C P18825 1/20 0.55
CCR2 P41597 1/20 0.55
CXCL12 P48061 1/20 0.55
BLM P54132 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
HRH3 Q9Y5N1 1/20 0.55
HTR6 P50406 1/20 0.53
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
ALOX15 P16050 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4741281 0.83 SIGMAR1 (0.54) TSHRMAPTCXCR4MEN1KMT2A
SCHEMBL4198058 0.80 CD4 (0.61) TSHRALDH1A1SMN1; SMN2
SCHEMBL722275 0.80 SIGMAR1 (0.56) CXCR4MEN1KMT2ACHRM2CHRM1
SCHEMBL614784 0.80 KDM4E (0.58) CXCR4MEN1KMT2ACHRM2CHRM1
SCHEMBL3969181 0.79 LMNA (0.62) TSHRALDH1A1SMN1; SMN2
SCHEMBL4786278 0.79 KMT2A (0.60) TSHRMAPTUSP2MEN1KMT2A
SCHEMBL19392254 0.78 TSHR (0.58) TSHRUSP2MEN1KMT2AHRH3
Hydrochloric Acid SCHEMBL29045124 0.78 CXCR4 (0.57) CXCR4MEN1KMT2ACHRM2CHRM1
Hydrochloric Acid SCHEMBL4786214 0.78 KMT2A (0.59) TSHRMAPTUSP2MEN1KMT2A
SCHEMBL6765737 0.78 CXCR4 (0.67) CXCR4MEN1KMT2ACHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO claimed
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO disclosed