SCHEMBL25522223

SCHEMBL25522223

Cc1ccc(CNCc2ncccc2C)nc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 1/20 0.39
ADORA2A P29274 6/20 0.38
ADORA1 P30542 5/20 0.38
HTR1A P08908 5/20 0.37
HTT P42858 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
IGF1R P08069 1/20 0.35
FGFR1 P11362 1/20 0.35
KDR P35968 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2A6 P11509 1/20 0.34
CHRM2 P08172 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
DYRK1B Q9Y463 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25523333 0.85 IGF1R (0.38) SCN8AADORA2AADORA1HTTIGF1R
SCHEMBL25523327 0.85 ADORA2A (0.41) ADORA2AHTR1ATLR7MAOAMAOB
SCHEMBL2082460 0.83 NOS3 (0.45) SCN8AADORA2AADORA1HTTIGF1R
SCHEMBL30481998 0.83 SCN8A (0.55) SCN8ACYP3A4CHRM2MAOAMAOB
SCHEMBL23775046 0.82 NPC1 (0.47) SCN8AMAOAMAOB
SCHEMBL25522228 0.81 TLR7 (0.41) SCN8AADORA2AHTR1ATLR7CHRM2
SCHEMBL2261106 0.75 NOS3 (0.41) ADORA2AADORA1IGF1RFGFR1KDR
SCHEMBL14477280 0.75 CCR1 (0.43) HTR1ACHRM2
SCHEMBL2084689 0.74 ADORA2A (0.44) ADORA2AADORA1HTTIGF1RFGFR1
SCHEMBL25378467 0.74 HTT (0.50) SCN8AADORA2AADORA1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230159510-A1 NOVEL PRMT5 INHIBITORS AMGEN INC. (US) 2023-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230159510-A1 NOVEL PRMT5 INHIBITORS PRMT5, PRMT1, PRMT3 SCN8A 4172/4885ADORA2A 4422/4885ADORA1 3747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.