SCHEMBL2552243

SCHEMBL2552243

CN(C)CCOC(C(=O)O)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 7/20 0.62
CHRM1 P11229 5/20 0.62
CHRM2 P08172 4/20 0.62
CYP2D6 P10635 4/20 0.62
ADRA2A P08913 3/20 0.62
SLC6A2 P23975 3/20 0.62
SLC6A4 P31645 3/20 0.62
OPRM1 P35372 3/20 0.62
DRD3 P35462 3/20 0.62
SLC6A3 Q01959 3/20 0.62
CHRM3 P20309 3/20 0.62
HTR2A P28223 3/20 0.62
HRH1 P35367 3/20 0.62
CHRM4 P08173 2/20 0.62
CHRM5 P08912 2/20 0.62
ADRA2B P18089 2/20 0.62
HRH2 P25021 2/20 0.62
HTR2C P28335 2/20 0.62
ADRA1A P35348 2/20 0.62
HTR2B P41595 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8833037 0.90 LMNA (0.62) LMNACHRM1CHRM2CYP2D6ADRA2A
SCHEMBL30728008 0.87 LMNA (0.58) LMNACHRM1CHRM2CYP2D6ADRA2A
SCHEMBL17724542 0.81 PPARA (0.47) LMNACYP2D6CYP1A2SMN1; SMN2CYP3A4
SCHEMBL8084866 0.81 PPARA (0.47) LMNACYP2D6CYP1A2SMN1; SMN2CYP3A4
Diphenhydramine SCHEMBL25268546 0.80 SLC6A2 (0.83) LMNACHRM1CHRM2CYP2D6ADRA2A
Diphenhydramine SCHEMBL25269204 0.80 SLC6A2 (0.83) LMNACHRM1CHRM2CYP2D6ADRA2A
SCHEMBL5831517 0.79 GLS (0.52) LMNACYP2D6CYP1A2TSHRCYP3A4
SCHEMBL21369008 0.79 GLS (0.50) LMNACYP2D6CYP1A2MAPK1CYP3A4
Diphenhydramine SCHEMBL29096592 0.79 LMNA (0.84) LMNACHRM1CHRM2CYP2D6ADRA2A
SCHEMBL21697916 0.78 LMNA (0.55) LMNACHRM1CHRM2CYP2D6ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed