SCHEMBL2549529

SCHEMBL2549529

O=C(O)N1Cc2cc(C3(Cl)CCC(c4ccc(F)cc4)CC3)ccc2-n2cnnc2C1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 5/20 0.35
OXTR P30559 4/20 0.33
AVPR1A P37288 2/20 0.31
HSD11B1 P28845 1/20 0.31
TACR1 P25103 1/20 0.30
KCNH2 Q12809 1/20 0.30
NAMPT P43490 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2552411 0.85 AVPR1A (0.34) AVPR1ATACR1KCNH2
SCHEMBL2564864 0.85 AVPR2 (0.37) AVPR2OXTRAVPR1AKCNH2
SCHEMBL2556524 0.82 CYP11B2 (0.32) AVPR2AVPR1AKCNH2
SCHEMBL2550063 0.81 NAMPT (0.40) AVPR2OXTRAVPR1ATACR1KCNH2
SCHEMBL2565565 0.81 AVPR1A (0.32) AVPR2OXTRAVPR1AKCNH2
SCHEMBL2564697 0.81 AVPR1A (0.31) AVPR2AVPR1AKCNH2
SCHEMBL2564173 0.81 AVPR2 (0.31) AVPR2
SCHEMBL2347000 0.81 AVPR2 (0.31) AVPR2OXTRAVPR1A
Hydrochloric Acid SCHEMBL2544777 0.80 AVPR1A (0.33) AVPR1A
SCHEMBL2549332 0.76 AVPR1A (0.37) AVPR2OXTRAVPR1AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552919-A1 ARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. Hoffmann-La Roche AG (CH) 2013-02-06 EP disclosed
WO-2011120877-A1 ARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-10-06 WO disclosed