SCHEMBL2552414

SCHEMBL2552414

CCN1CCC(NS(=O)(=O)c2ccc(CN3CCCC3C)cc2)C1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 14/20 0.55
KCNH2 Q12809 12/20 0.55
HTT P42858 1/20 0.47
THRB P10828 1/20 0.47
ALDH1A1 P00352 1/20 0.46
HRH2 P25021 1/20 0.44
HRH1 P35367 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2547933 0.81 KDM4E (0.48) HRH3KCNH2HTTTHRBALDH1A1
SCHEMBL2555109 0.81 KDM4E (0.48) HRH3KCNH2HTTTHRBALDH1A1
SCHEMBL7716908 0.81 KDM4E (0.48) HRH3KCNH2HTTTHRBALDH1A1
Hydrochloric Acid SCHEMBL2552429 0.80 KDM4E (0.47) HRH3KCNH2HTTTHRBALDH1A1
Hydrochloric Acid SCHEMBL2552428 0.80 KDM4E (0.47) HRH3KCNH2HTTTHRBALDH1A1
SCHEMBL2555154 0.79 KDM4E (0.48) HRH3KCNH2HTTALDH1A1
SCHEMBL11815516 0.78 KDM4E (0.49) HRH3KCNH2HTTALDH1A1
Hydrochloric Acid SCHEMBL9796292 0.78 ALDH1A1 (0.55) HTTTHRBALDH1A1HRH2HRH1
SCHEMBL2552379 0.76 HRH3 (0.45) HRH3KCNH2HTTTHRBALDH1A1
SCHEMBL2549964 0.76 KCNH2 (0.49) HRH3KCNH2HTTTHRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO disclosed
WO-2011121309-A1 PHENYL SULFONYL DERIVATIVES AND THEIR USE AS HISTAMINE H3 ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-10-06 WO disclosed