SCHEMBL25528176

SCHEMBL25528176

COc1cccc(CN2C(=O)c3ccc(-c4ccncc4)cc3N(C)C(=O)[C@H]2C)c1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 13/20 0.57
ROCK1 Q13464 10/20 0.57
TNIK Q9UKE5 3/20 0.46
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
PRKACA P17612 1/20 0.42
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
PRKX P51817 1/20 0.42
PRKCQ Q04759 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
AURKA O14965 1/20 0.41
HCRTR1 O43613 2/20 0.41
HCRTR2 O43614 2/20 0.41
CMA1 P23946 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528179 1.00 ROCK2 (0.57) ROCK2ROCK1TNIKCYP3A4CYP2D6
SCHEMBL25528180 0.89 ROCK2 (0.59) ROCK2ROCK1TNIKCYP3A4PRKACA
SCHEMBL25528181 0.89 ROCK2 (0.59) ROCK2ROCK1TNIKCYP3A4PRKACA
SCHEMBL25529500 0.85 ROCK2 (0.59) ROCK2ROCK1TNIKGSK3B
SCHEMBL25529501 0.84 ROCK1 (0.47) ROCK2ROCK1
SCHEMBL25531869 0.83 ROCK2 (0.42) ROCK2ROCK1TNIKCYP3A4CYP2D6
SCHEMBL29249878 0.80 ROCK2 (0.62) ROCK2ROCK1TNIKCYP3A4CYP2D6
SCHEMBL30914656 0.80 ROCK2 (0.62) ROCK2ROCK1TNIKCYP3A4CYP2D6
SCHEMBL25528471 0.79 ROCK2 (0.44) ROCK2ROCK1HCRTR1HCRTR2
SCHEMBL30914662 0.77 ROCK2 (0.69) ROCK2ROCK1TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed