SCHEMBL25528181

SCHEMBL25528181

COc1cccc(CN2C(=O)c3ccc(-c4ccnc(N)c4)cc3N(C)C(=O)[C@H]2C)c1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.59
ROCK1 Q13464 7/20 0.59
TNIK Q9UKE5 7/20 0.47
CYP3A4 P08684 2/20 0.43
PRKACA P17612 2/20 0.43
DYRK1A Q13627 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528180 1.00 ROCK2 (0.59) ROCK2ROCK1TNIKCYP3A4PRKACA
SCHEMBL25528176 0.89 ROCK2 (0.57) ROCK2ROCK1TNIKCYP3A4PRKACA
SCHEMBL25528179 0.89 ROCK2 (0.57) ROCK2ROCK1TNIKCYP3A4PRKACA
SCHEMBL25528328 0.82 BRD4 (0.43) ROCK2ROCK1CYP3A4
SCHEMBL25529357 0.81 ROCK2 (0.65) ROCK2ROCK1TNIKCYP3A4PRKACA
SCHEMBL25528184 0.81 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25528333 0.80 ROCK2 (0.39) ROCK2ROCK1PRKACA
SCHEMBL25528187 0.80 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25528190 0.80 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25528332 0.79 ROCK2 (0.38) ROCK2ROCK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed