SCHEMBL25529501

SCHEMBL25529501

C[C@@H]1C(=O)N(C)c2cc(-c3ccncc3)ccc2C(=O)N1Cc1cccc(C(=O)O)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 7/20 0.47
ROCK2 O75116 7/20 0.47
KMT2A Q03164 1/20 0.41
PRKAG1 P54619 2/20 0.39
PRKAA2 P54646 2/20 0.39
PRKAB1 Q9Y478 2/20 0.39
IDO1 P14902 2/20 0.39
TDO2 P48775 1/20 0.39
BRD4 O60885 1/20 0.38
HTT P42858 1/20 0.38
CYP19A1 P11511 1/20 0.38
KDM4A O75164 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25530887 0.90 KMT2A (0.39) ROCK1ROCK2KMT2APRKAG1PRKAA2
SCHEMBL25529500 0.90 ROCK2 (0.59) ROCK1ROCK2IDO1BRD4
SCHEMBL25528471 0.87 ROCK2 (0.44) ROCK1ROCK2IDO1TDO2BRD4
SCHEMBL25530907 0.84 IRAK4 (0.43) ROCK1ROCK2BRD4
SCHEMBL25528176 0.84 ROCK2 (0.57) ROCK1ROCK2
SCHEMBL25528179 0.84 ROCK2 (0.57) ROCK1ROCK2
SCHEMBL25528185 0.84 ROCK2 (0.43) ROCK1ROCK2
SCHEMBL25529068 0.84 ROCK2 (0.43) ROCK1ROCK2
SCHEMBL25530880 0.80 ROCK1 (0.48) ROCK1ROCK2KMT2AIDO1
SCHEMBL25530634 0.79 ROCK2 (0.40) ROCK1ROCK2KMT2APRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed