SCHEMBL25528351

SCHEMBL25528351

CN/C(=C(/C)C=N)c1ccc2c(c1)N(C)C(=O)[C@@H](C)N(Cc1cccc(C(=O)NCC3(O)CC3)c1)C2=O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.34
THRB P10828 1/20 0.33
CACNA1G O43497 7/20 0.33
NAMPT P43490 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RIPK1 Q13546 1/20 0.32
GAA P10253 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
DRD2 P14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528758 0.86 PARP1 (0.42) BRD4THRBCACNA1GNAMPT
SCHEMBL25528350 0.84 BRD4 (0.33) BRD4THRBCACNA1GGAANPSR1
SCHEMBL25528337 0.77 BRD4 (0.39) BRD4THRBCACNA1GALDH1A1GAA
SCHEMBL25528767 0.76 MAP4K4 (0.38) BRD4CACNA1GNAMPTGAA
SCHEMBL25528339 0.74 PARP1 (0.41) BRD4THRBCACNA1GNAMPT
SCHEMBL25528752 0.74 PARP1 (0.42) BRD4THRBCACNA1GNAMPT
SCHEMBL25528749 0.69 IRAK4 (0.41)
SCHEMBL25528328 0.68 BRD4 (0.43) BRD4
SCHEMBL25528200 0.67 ROCK2 (0.40)
SCHEMBL25529498 0.66 MAPT (0.48) THRBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed