SCHEMBL25528328

SCHEMBL25528328

CCNC(=O)c1cccc(CN2C(=O)c3ccc(-c4ccnc(N)c4)cc3N(C)C(=O)[C@H]2C)c1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.43
ROCK2 O75116 12/20 0.40
ROCK1 Q13464 7/20 0.40
CYP3A4 P08684 1/20 0.35
CYP3A5 P20815 1/20 0.35
DPP4 P27487 1/20 0.34
AOC3 Q16853 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528333 0.92 ROCK2 (0.39) BRD4ROCK2ROCK1
SCHEMBL25528200 0.91 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25528201 0.90 ROCK2 (0.39) ROCK2ROCK1
SCHEMBL25528196 0.88 ROCK2 (0.43) BRD4ROCK2ROCK1
SCHEMBL25528332 0.88 ROCK2 (0.38) ROCK2ROCK1CYP3A4
SCHEMBL25528334 0.87 NPSR1 (0.45) ROCK2ROCK1
SCHEMBL25529692 0.84 ROCK2 (0.52) ROCK2ROCK1
SCHEMBL25528651 0.83 ROCK2 (0.38) BRD4ROCK2ROCK1
SCHEMBL25529691 0.83 ROCK2 (0.40) BRD4ROCK2ROCK1
SCHEMBL25528181 0.82 ROCK2 (0.59) ROCK2ROCK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed