SCHEMBL25528474

SCHEMBL25528474

Cc1ccc(C(=O)OC2CN(C(=O)c3cccc(CN4C(=O)c5ccc(-c6ccncc6)cc5N(C)C(=O)[C@H]4C)c3)C2)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.41
ROCK1 Q13464 4/20 0.41
CYP46A1 Q9Y6A2 7/20 0.36
BRD4 O60885 1/20 0.34
TAF1 P21675 1/20 0.34
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
CYP3A4 P08684 1/20 0.33
BACE1 P56817 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528750 0.91 ROCK2 (0.33) ROCK2ROCK1CYP46A1BRD4GRIN2B
SCHEMBL25528189 0.86 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25532225 0.86 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25528471 0.84 ROCK2 (0.44) ROCK2ROCK1CYP46A1BRD4TAF1
SCHEMBL25528478 0.82 ROCK2 (0.41) ROCK2ROCK1CYP46A1BRD4
SCHEMBL25529500 0.80 ROCK2 (0.59) ROCK2ROCK1BRD4IDO1
SCHEMBL25529070 0.79 CACNA1H (0.33) ROCK2ROCK1BRD4
SCHEMBL25532515 0.79 ROCK2 (0.33) ROCK2ROCK1BRD4
SCHEMBL25528479 0.79 CACNA1H (0.33) ROCK2ROCK1BRD4
SCHEMBL25529501 0.79 ROCK1 (0.47) ROCK2ROCK1BRD4IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed