SCHEMBL25528619

SCHEMBL25528619

Cc1cc(F)cc(C(=O)OC2CC(CNC(=O)c3cccc(CN4C(=O)c5ccc(-c6ccncc6)cc5N(C)C(=O)[C@H]4C)c3)C2)c1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 17/20 0.40
ROCK1 Q13464 7/20 0.40
AURKA O14965 2/20 0.35
CACNA1H O95180 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528924 0.94 CACNA1H (0.37) ROCK2ROCK1AURKACACNA1H
SCHEMBL25528189 0.89 ROCK2 (0.40) ROCK2ROCK1
SCHEMBL25532600 0.89 CACNA1H (0.33) ROCK2ROCK1AURKACACNA1H
SCHEMBL25529081 0.88 ROCK2 (0.36) ROCK2ROCK1AURKACACNA1H
SCHEMBL25529087 0.88 ROCK2 (0.34) ROCK2ROCK1AURKACACNA1H
SCHEMBL25528480 0.87 ROCK2 (0.43) ROCK2ROCK1
SCHEMBL25530084 0.87 ROCK2 (0.41) ROCK2ROCK1AURKA
SCHEMBL25528921 0.87 ROCK2 (0.41) ROCK2ROCK1AURKA
SCHEMBL25528185 0.85 ROCK2 (0.43) ROCK2ROCK1AURKA
SCHEMBL25529068 0.85 ROCK2 (0.43) ROCK2ROCK1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed