SCHEMBL25528844

SCHEMBL25528844

C[C@@H]1C(=O)N(C)c2cc(-c3ccncc3)ccc2C(=O)N1Cc1cccc(C(=O)NCC2(COC(=O)c3ccc(Cl)c(Cl)c3)CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 16/20 0.42
ROCK1 Q13464 6/20 0.42
AURKA O14965 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
PRKACA P17612 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
PRKX P51817 1/20 0.32
PRKCQ Q04759 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25528615 0.91 ROCK1 (0.34) ROCK2ROCK1AURKAALDH1A1
SCHEMBL25528842 0.86 ROCK2 (0.41) ROCK2ROCK1AURKAALDH1A1CYP3A4
SCHEMBL25528480 0.85 ROCK2 (0.43) ROCK2ROCK1
SCHEMBL25531869 0.81 ROCK2 (0.42) ROCK2ROCK1ALDH1A1CYP3A4CYP2D6
SCHEMBL25529500 0.80 ROCK2 (0.59) ROCK2ROCK1GSK3B
SCHEMBL25528837 0.80 ROCK2 (0.32) ROCK2ROCK1
SCHEMBL25528478 0.79 ROCK2 (0.41) ROCK2ROCK1AURKA
SCHEMBL25529068 0.77 ROCK2 (0.43) ROCK2ROCK1AURKA
SCHEMBL25528185 0.77 ROCK2 (0.43) ROCK2ROCK1AURKA
SCHEMBL25529501 0.76 ROCK1 (0.47) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed