SCHEMBL25530645

SCHEMBL25530645

COC(=O)c1cccc(CN(CC=O)C(=O)c2ccc(Br)cc2N(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 2/20 0.43
CYP4A11 Q02928 2/20 0.43
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
CCR5 P51681 1/20 0.40
SLC7A5 Q01650 1/20 0.39
NR3C1 P04150 1/20 0.38
MAPK8 P45983 1/20 0.37
LMNA P02545 2/20 0.37
MEP1B Q16820 1/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
CASR P41180 1/20 0.36
MRGPRX4 Q96LA9 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
PTGES O14684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25530657 0.81 ROCK2 (0.38) CYP4F2CYP4A11KDM4EALDH1A1MAPT
SCHEMBL3124357 0.78 LOXL2 (0.55) CYP4F2CYP4A11KDM4EALDH1A1MAPT
SCHEMBL12393362 0.73 LOXL2 (0.48) CYP4F2CYP4A11KDM4EALDH1A1MAPT
SCHEMBL25530669 0.70 AOC3 (0.36) LOXL2MEP1BKMT2AMRGPRX4L3MBTL1
SCHEMBL4813988 0.70 NR4A2 (0.49) KDM4EALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL165622 0.69 LOXL2 (0.66) CYP4F2CYP4A11KDM4EALDH1A1MAPT
SCHEMBL31565671 0.68 NR4A2 (0.47) KDM4EALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL697890 0.68 LOXL2 (0.68) CYP4F2CYP4A11KDM4EALDH1A1MAPT
SCHEMBL31753372 0.66 CYP4A11 (0.72) CYP4F2CYP4A11KDM4EALDH1A1MAPT
SCHEMBL28212 0.66 LOXL2 (0.70) CYP4F2CYP4A11KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed