SCHEMBL2553564

SCHEMBL2553564

CCN(C(=O)O)c1ccc(Br)cc1F

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 2/20 0.44
DGAT1 O75907 1/20 0.41
FPR2 P25090 1/20 0.39
TMEM97 Q5BJF2 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
ALDH1A1 P00352 5/20 0.38
MAPT P10636 3/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
POLB P06746 1/20 0.37
LMNA P02545 3/20 0.37
NPC1 O15118 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NR2F2 P24468 1/20 0.36
GLA P06280 1/20 0.36
TSHR P16473 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086382 0.81 PTK2 (0.43) PTK2DGAT1TMEM97SIGMAR1ALDH1A1
SCHEMBL2552329 0.80 AAK1 (0.42) PTK2DGAT1FPR2ALDH1A1MAPT
SCHEMBL17420936 0.78 SIRT2 (0.48) PTK2DGAT1TMEM97SIGMAR1ALDH1A1
SCHEMBL17078095 0.76 TSHR (0.48) SIGMAR1ALDH1A1MAPTLMNAGLA
SCHEMBL6832796 0.75 ALDH1A1 (0.44) DGAT1ALDH1A1MAPTSIRT2THRB
SCHEMBL3991292 0.75 DGAT1 (0.42) PTK2DGAT1FPR2TMEM97SIGMAR1
SCHEMBL57513 0.74 DGAT1 (0.41) PTK2DGAT1FPR2TMEM97SIGMAR1
SCHEMBL3892297 0.74 DPP4 (0.35) PTK2DGAT1ALDH1A1SIRT2LMNA
SCHEMBL3892298 0.74 DPP4 (0.35) PTK2DGAT1ALDH1A1SIRT2LMNA
SCHEMBL27906114 0.72 AAK1 (0.40) PTK2DGAT1FPR2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552206-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-02-06 EP disclosed
WO-2011123419-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2011-10-06 WO disclosed