SCHEMBL255371

SCHEMBL255371

O=C(Nc1ccc2[nH]nc(C3C=CN=CC3)c2c1)C1CNCC(c2ccccc2)C1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 16/20 0.45
PDPK1 O15530 1/20 0.39
ITK Q08881 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL173378 0.78 ULK1 (0.49) ULK1PDPK1ITK
SCHEMBL12073259 0.67 KDM4E (0.40) PDPK1ITK
SCHEMBL18197025 0.66 NAMPT (0.39) ULK1
SCHEMBL23390296 0.64 LIPE (0.52)
Hydrochloric Acid SCHEMBL23390063 0.63 LIPE (0.51)
Hydrochloric Acid SCHEMBL23390064 0.63 LIPE (0.51)
SCHEMBL15043259 0.62 KHK (0.39) ULK1PDPK1
SCHEMBL486433 0.62 F2R (0.59)
SCHEMBL5594098 0.61 AURKA (0.68)
SCHEMBL4008398 0.61 AKR1C3 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012030685-A2 INDAZOLE DERIVATIVES USEFUL AS ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-08 WO disclosed