SCHEMBL2554451

SCHEMBL2554451

CN(C)Cc1ccc(B(O)O)cc1S(C)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.43
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
SLC6A4 P31645 4/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
G6PD P11413 1/20 0.35
PABPC1 P11940 1/20 0.35
HKDC1 Q2TB90 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2553161 0.82 ENPP2 (0.47) ENPP2CA2PTGS2
SCHEMBL30816185 0.76 ENPP2 (0.34) ENPP2CYP2C19CYP1A2ALDH1A1MEN1
SCHEMBL27159787 0.76 ENPP2 (0.34) ENPP2CYP2C19CYP1A2ALDH1A1MEN1
SCHEMBL2555834 0.76 CCR5 (0.42) CYP2C19CYP1A2SLC6A4KMT2AGAA
SCHEMBL19214301 0.75 ENPP2 (0.50) ENPP2CA2
SCHEMBL30643101 0.73 TTR (0.46) ENPP2CYP2C19CYP1A2SLC6A4ALDH1A1
SCHEMBL30643134 0.73 KDM4E (0.44) CYP2C19CYP1A2SLC6A4ALDH1A1MEN1
SCHEMBL2552371 0.73 SLC6A4 (0.39) CYP2C19CYP1A2SLC6A4ALDH1A1MEN1
SCHEMBL4010773 0.73 ENPP2 (0.52) ENPP2ALDH1A1GAAL3MBTL1CA2
SCHEMBL24804602 0.73 HSD17B10 (0.41) ENPP2SLC6A4ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed