SCHEMBL2554880

SCHEMBL2554880

O=C(O)N(Br)c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.46
TSHR P16473 2/20 0.46
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 2/20 0.43
HSD17B10 Q99714 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
SRD5A2 P31213 1/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP3A4 P08684 1/20 0.41
GSK3B P49841 1/20 0.40
CASP1 P29466 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CYP2C19 P33261 2/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3042400 0.80 NPSR1 (0.50) ALOX15TSHRALDH1A1SMN1; SMN2NPC1
SCHEMBL1703981 0.79 ALDH1A1 (0.44) TSHRALDH1A1SMN1; SMN2MAPTRAB9A
SCHEMBL692996 0.79 ALDH1A1 (0.48) ALOX15TSHRALDH1A1SMN1; SMN2MAPT
Hydrochloric Acid SCHEMBL11842627 0.77 ALDH1A1 (0.47) ALOX15TSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL1006640 0.77 HTR3E (0.43) TSHRALDH1A1SMN1; SMN2MAPTNPC1
SCHEMBL6129408 0.76 ALDH1A1 (0.56) ALOX15TSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL3953896 0.74 ALOX15 (0.44) ALOX15TSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL18605308 0.74 ALDH1A1 (0.44) ALOX15TSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL2096920 0.73 NPSR1 (0.54) ALOX15TSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL11176346 0.73 ALDH1A1 (0.43) ALOX15TSHRALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2558069-A1 BENZONAPTHYRIDINE COMPOSITIONS AND USES THEREOF Novartis AG (CH) 2013-02-20 EP disclosed
WO-2011130379-A1 BENZONAPTHYRIDINE COMPOSITIONS AND USES THEREOF NOVARTIS AG (CH) 2011-10-20 WO disclosed