SCHEMBL2554963

SCHEMBL2554963

CC(C)=CCCC(C)C(C)=CC=O

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.48
TSHR P16473 1/20 0.48
ALDH1A1 P00352 3/20 0.48
USP2 O75604 1/20 0.34
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
SRC P12931 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2554959 1.00 ALOX15 (0.48) ALOX15TSHRALDH1A1USP2GLA
SCHEMBL11454435 0.79 ALDH1A1 (0.42) ALOX15TSHRALDH1A1
SCHEMBL11454436 0.79 ALDH1A1 (0.42) ALOX15TSHRALDH1A1
SCHEMBL1784816 0.77 FDPS (0.34) TSHRALDH1A1
SCHEMBL1784814 0.77 FDPS (0.34) TSHRALDH1A1
SCHEMBL6050618 0.75 ALOX15 (0.52) ALOX15TSHRALDH1A1USP2GLA
SCHEMBL11869803 0.74 ALOX15 (0.50) ALOX15TSHRALDH1A1USP2GLA
SCHEMBL28167129 0.74 ALOX15 (0.50) ALOX15TSHRALDH1A1USP2GLA
SCHEMBL1787529 0.73 CA1 (0.41) TSHR
SCHEMBL1787528 0.73 CA1 (0.41) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-9554990-B2 Cholecystokinin secretion-promoting composition J-OIL MILLS, INC. (JP) 2017-01-31 US disclosed
US-20160106668-A1 CHOLECYSTOKININ SECRETION-PROMOTING COMPOSITION J-OIL MILLS, INC. (JP) 2016-04-21 US disclosed
US-20150164823-A1 CHOLECYSTOKININ SECRETION-PROMOTING COMPOSITION J-OIL MILLS, INC. (JP) 2015-06-18 US disclosed
CN-104661659-A Cholecystokinin secretion-promoting composition J OIL MILLS INC 2015-05-27 CN disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed