SCHEMBL2555372

SCHEMBL2555372

O=Cc1c[nH]c(-c2ccc(F)c(F)c2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMP P19971 1/20 0.41
GRK6 P43250 1/20 0.38
KMO O15229 2/20 0.37
NOTUM Q6P988 1/20 0.37
TERT O14746 1/20 0.36
CYP17A1 P05093 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
ALDH1A1 P00352 2/20 0.34
IDO1 P14902 1/20 0.34
CYP1A2 P05177 1/20 0.34
GAA P10253 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
DYRK1A Q13627 1/20 0.34
MAOB P27338 1/20 0.33
KCNH2 Q12809 1/20 0.33
ERN1 O75460 1/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2558891 0.86 ESR1 (0.45) GRK6CYP17A1CYP11B1CYP11B2ERN1
SCHEMBL2560329 0.86 ERN1 (0.43) TYMPKMOGAAERN1
SCHEMBL15332262 0.86 DAPK3 (0.38) DYRK1AMEN1KMT2ARAB9A
SCHEMBL15331416 0.86 KMO (0.41) KMOTERTMAOB
SCHEMBL15329600 0.86 ERCC1 (0.43) KMO
SCHEMBL2557559 0.86 PARP1 (0.36) TYMPMAOB
SCHEMBL2563031 0.83 LRRK2 (0.39) CYP11B1CYP11B2
SCHEMBL15329643 0.83 ERN1 (0.47) CYP17A1ALDH1A1GAAERN1PDGFRB
SCHEMBL15330812 0.82 ALDH1A1 (0.42) ALDH1A1CYP1A2GAACYP2C19ERN1
SCHEMBL15332789 0.81 KDM4E (0.38) TYMPTERTALDH1A1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed