SCHEMBL2555759

SCHEMBL2555759

CS(=O)(=O)c1ccc(Br)c(C=O)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.44
PRKDC P78527 1/20 0.41
ENPP2 Q13822 2/20 0.39
G6PD P11413 1/20 0.39
IDE P14735 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PTGS2 P35354 3/20 0.38
LMNA P02545 2/20 0.38
EPAS1 Q99814 1/20 0.37
PTGS1 P23219 1/20 0.37
SIRT1 Q96EB6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31733573 0.86 PRKDC (0.44) ERN1PRKDCENPP2G6PDIDE
SCHEMBL7857418 0.81 HTT (0.42) ERN1PRKDCSMN1; SMN2PTGS2LMNA
SCHEMBL26777577 0.80 ALDH1A1 (0.41) ERN1PRKDCSMN1; SMN2LMNA
SCHEMBL20083904 0.80 ERN1 (0.44) ERN1ENPP2G6PDIDESMN1; SMN2
SCHEMBL136274 0.78 ERN1 (0.53) ERN1ENPP2
SCHEMBL21491267 0.78 LMNA (0.51) ERN1PTGS2LMNA
SCHEMBL7752223 0.78 PTGS2 (0.48) ERN1PTGS2PTGS1
SCHEMBL12593470 0.76 SMN1; SMN2 (0.52) ERN1ENPP2G6PDIDESMN1; SMN2
SCHEMBL15814013 0.76 ALDH1A1 (0.43) ERN1ENPP2G6PDIDESMN1; SMN2
SCHEMBL7092074 0.76 SMN1; SMN2 (0.61) ERN1PRKDCSMN1; SMN2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621135-B LPA1 small molecule antagonist 上海拓界生物医药科技有限公司 2024-01-30 CN disclosed
CN-114621135-A LPA1 small molecule antagonist 上海拓界生物医药科技有限公司 2022-06-14 CN disclosed
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed