SCHEMBL25565477

SCHEMBL25565477

CC(C)C(=O)N1CCC(CN2CN(C(C)C)C2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.38
KCNH2 Q12809 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37
RORC P51449 1/20 0.36
HTR4 Q13639 2/20 0.36
CYP2D6 P10635 1/20 0.36
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
XBP1 P17861 1/20 0.35
MAPK1 P28482 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
THRB P10828 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
CHRNB3 Q05901 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25558120 0.91 HRH3 (0.39) FAAHKCNH2HRH3L3MBTL1MEN1
SCHEMBL22520608 0.88 HRH3 (0.44) FAAHKCNH2HRH3L3MBTL1MEN1
SCHEMBL24669824 0.84 CACNA2D1 (0.41) FAAHKCNH2HRH3ALDH1A1CYP2D6
SCHEMBL25558060 0.84 CHRNB2 (0.43) KCNH2CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL27425177 0.83 CACNA2D1 (0.45) FAAHL3MBTL1MEN1ALDH1A1KMT2A
SCHEMBL25558598 0.82 KCNH2 (0.38) FAAHKCNH2HRH3HTR4CYP2D6
SCHEMBL12413703 0.82 MAPT (0.48) TP53THRBMAPT
SCHEMBL25551823 0.80 KCNH2 (0.40) KCNH2HRH3HTR4CYP2D6EPHX2
SCHEMBL25560580 0.79 HRH3 (0.39) KCNH2HRH3HTR4NPSR1
SCHEMBL22520730 0.79 HSD11B1 (0.41) FAAHL3MBTL1MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023096995-A1 COMPOSITIONS AND METHODS COMPRISING SUBSTITUTED N-(2-CHLORO-6-METHYLPHENYL)-2-((6-(6-MEMBERED HETEROCYCLOALKYL)-2-METHYLPYRIMIDIN-4-YL)AMINO)THIAZOLE-5-CARBOXAMIDE ANALOGUES ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2023-06-01 WO disclosed