SCHEMBL25566965

SCHEMBL25566965

O=C(O)CC12CCC(CN(Cc3ccccc3)C1)N2Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 5/20 0.43
CHRM2 P08172 4/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
S1PR1 P21453 1/20 0.41
S1PR5 Q9H228 1/20 0.41
GAA P10253 1/20 0.40
FAAH O00519 1/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25566966 0.87 CYP2D6 (0.42) CHRM3CHRM2ALDH1A1GAABCHE
SCHEMBL25566734 0.85 FUCA1 (0.42) CHRM3CHRM2ALDH1A1
SCHEMBL25566962 0.80 ACHE (0.39) CHRM3CHRM2MEN1KMT2AALDH1A1
SCHEMBL25566963 0.80 KDM1A (0.47) CHRM3CHRM2
SCHEMBL25566735 0.79 ACHE (0.38) CHRM3CHRM2GAAACHE
SCHEMBL29937525 0.79 CHRM3 (0.42) CHRM3CHRM2MEN1KMT2AALDH1A1
SCHEMBL29937437 0.78 CHRM3 (0.41) CHRM3CHRM2MEN1KMT2AALDH1A1
SCHEMBL31091663 0.77 CYP2D6 (0.42) CHRM3CHRM2MEN1KMT2ATSHR
SCHEMBL29936728 0.72 KMT2A (0.43) CHRM3CHRM2KMT2AALDH1A1MAPT
SCHEMBL29344022 0.72 KMT2A (0.43) CHRM3CHRM2KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4442686-A1 KRAS INHIBITORS, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF Abbisko Therapeutics Co., Ltd (CN) 2024-10-09 EP disclosed
CN-118055932-A KRAS inhibitor and preparation and pharmaceutical application thereof 上海和誉生物医药科技有限公司 2024-05-17 CN disclosed
WO-2023098425-A1 KRAS INHIBITORS, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 上海和誉生物医药科技有限公司 2023-06-08 WO disclosed