SCHEMBL25566966

SCHEMBL25566966

COC(=O)CC12CCC(CN(Cc3ccccc3)C1)N2Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.42
ALDH1A1 P00352 1/20 0.42
BCHE P06276 3/20 0.40
MAOB P27338 2/20 0.40
ACHE P22303 2/20 0.40
NR1H2 P55055 1/20 0.40
CHRM2 P08172 2/20 0.39
CHRM3 P20309 2/20 0.39
GAA P10253 1/20 0.39
MCHR1 Q99705 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25566965 0.87 CHRM3 (0.43) ALDH1A1BCHEACHECHRM2CHRM3
SCHEMBL25566962 0.82 ACHE (0.39) CYP2D6ALDH1A1ACHECHRM2CHRM3
SCHEMBL25566734 0.80 FUCA1 (0.42) ALDH1A1CHRM2CHRM3
SCHEMBL25566735 0.79 ACHE (0.38) ACHECHRM2CHRM3GAA
SCHEMBL31091663 0.77 CYP2D6 (0.42) CYP2D6ALDH1A1ACHECHRM2CHRM3
SCHEMBL29937525 0.76 CHRM3 (0.42) CYP2D6ALDH1A1BCHEACHECHRM2
SCHEMBL29937437 0.75 CHRM3 (0.41) CYP2D6ALDH1A1CHRM2CHRM3GAA
SCHEMBL25566963 0.75 KDM1A (0.47) CHRM2CHRM3SIGMAR1
SCHEMBL30998665 0.73 KMT2A (0.42) CYP2D6ALDH1A1CHRM2CHRM3
SCHEMBL29936728 0.73 KMT2A (0.43) CYP2D6ALDH1A1BCHEACHECHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4442686-A1 KRAS INHIBITORS, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF Abbisko Therapeutics Co., Ltd (CN) 2024-10-09 EP disclosed
WO-2023098425-A1 KRAS INHIBITORS, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 上海和誉生物医药科技有限公司 2023-06-08 WO disclosed