SCHEMBL25604262

SCHEMBL25604262

CC(C)(C)OC(=O)N1CCc2c(ccc3c(CC(=O)O)noc23)C1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.46
NR1H2 P55055 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.41
SCN9A Q15858 1/20 0.40
UCHL1 P09936 1/20 0.39
ACACB O00763 1/20 0.39
ADORA1 P30542 2/20 0.39
MAPK1 P28482 1/20 0.38
MAPT P10636 3/20 0.37
P2RX3 P56373 1/20 0.37
F12 P00748 2/20 0.36
KDM4E B2RXH2 1/20 0.36
PARP1 P09874 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
LIPG Q9Y5X9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25604354 0.93 SMN1; SMN2 (0.42) ESR2NR1H2SMN1; SMN2ADORA1MAPT
SCHEMBL25604198 0.92 ESR2 (0.46) ESR2NR1H2SMN1; SMN2SCN9AADORA1
SCHEMBL25825901 0.91 SMN1; SMN2 (0.44) ESR2NR1H2SMN1; SMN2MAPK1MAPT
SCHEMBL25604356 0.82 ESR2 (0.39) ESR2NR1H2SMN1; SMN2ADORA1
SCHEMBL25604199 0.81 ESR2 (0.43) ESR2NR1H2SMN1; SMN2ADORA1MAPK1
SCHEMBL25825839 0.80 SMN1; SMN2 (0.40) NR1H2SMN1; SMN2MAPTPARP1
SCHEMBL25825902 0.79 L3MBTL1 (0.39) ESR2NR1H2SMN1; SMN2ADORA1MAPK1
SCHEMBL25604141 0.75 MAPT (0.46) ESR2NR1H2SMN1; SMN2MAPK1MAPT
SCHEMBL25604260 0.72 ESR2 (0.54) ESR2NR1H2SCN9AUCHL1ACACB
SCHEMBL2117366 0.71 ESR2 (0.61) ESR2NR1H2SCN9AUCHL1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125944-A1 COMPOUND CONTAINING HETEROCYCLIC RING 正大天晴药业集团股份有限公司 2023-07-06 WO disclosed
WO-2023088406-A1 FUSED IMIDE DERIVATIVE 正大天晴药业集团股份有限公司 2023-05-25 WO disclosed