SCHEMBL2560682

SCHEMBL2560682

N#Cc1cncc(Cc2cncc(C#N)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
HRH3 Q9Y5N1 2/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
RAF1 P04049 1/20 0.38
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
HTT P42858 1/20 0.35
CHRNB2 P17787 4/20 0.35
CHRNA4 P43681 4/20 0.35
CHRNB4 P30926 3/20 0.35
CHRNA3 P32297 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27402031 0.89 ADORA1 (0.49) ADORA2AADORA1HRH3CYP11B1CYP11B2
SCHEMBL31739220 0.89 ADORA1 (0.49) ADORA2AADORA1HRH3CYP11B1CYP11B2
SCHEMBL16619272 0.84 LOXL2 (0.52) HRH3RAF1
SCHEMBL1413347 0.83 LOXL2 (0.48) ADORA2AADORA1HRH3CYP11B1CYP11B2
SCHEMBL7673123 0.83 CYP11B1 (0.38) ADORA2AADORA1HRH3CYP11B1CYP11B2
SCHEMBL29625378 0.83 CYP11B1 (0.38) ADORA2AADORA1HRH3CYP11B1CYP11B2
SCHEMBL1161457 0.83 CYP11B1 (0.38) ADORA2AADORA1HRH3CYP11B1CYP11B2
SCHEMBL19911768 0.83 CYP11B2 (0.47) ADORA2AADORA1HRH3CYP11B1CYP11B2
SCHEMBL1413419 0.83 GRIN2B (0.40) HRH3CYP11B1CYP11B2RAF1GRIN1
SCHEMBL1413439 0.83 CYP11B1 (0.47) ADORA2AADORA1HRH3CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011130741-A1 COMPOUNDS FOR TREATING NEURODEGENERATIVE DISEASES ARRAY BIOPHARMA INC. (US) 2011-10-20 WO disclosed