SCHEMBL256086

SCHEMBL256086

CCc1ccc(C#Cc2ccccc2Cl)o1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.44
GRM5 P41594 2/20 0.41
PTGDR2 Q9Y5Y4 6/20 0.38
FFAR1 O14842 1/20 0.36
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.31
PKM P14618 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL256077 0.82 GRM5 (0.38) GRM5PTGDR2PRSS1PRSS2PRSS3
SCHEMBL9967677 0.77 KCNH2 (0.44) KCNH2GRM5PTGDR2FFAR1PRSS1
SCHEMBL2108691 0.76 KCNH2 (0.42) KCNH2GRM5PTGDR2FFAR1PRSS1
SCHEMBL256660 0.75 KCNH2 (0.39) KCNH2GRM5PTGDR2ALDH1A1
SCHEMBL4448140 0.73 KCNH2 (0.61) KCNH2GRM5PTGDR2FFAR1ALDH1A1
SCHEMBL30707788 0.73 KCNH2 (0.61) KCNH2GRM5PTGDR2FFAR1ALDH1A1
SCHEMBL2108693 0.72 KCNH2 (0.39) KCNH2GRM5PTGDR2FFAR1PRSS1
SCHEMBL2637393 0.71 ALDH1A1 (0.50) PTGDR2FFAR1PRSS1PRSS2PRSS3
SCHEMBL15978536 0.70
SCHEMBL256672 0.69 GRM5 (0.39) KCNH2GRM5FFAR1PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028578-A1 SUBSTITUTED FUSED PYRIMIDINONES AND DIHYDROPYRIMIDINONES BAYER CROPSCIENCE AG (DE) 2012-03-08 WO disclosed