SCHEMBL2560955

SCHEMBL2560955

CC(C)CCC1CCc2ccc(OC3CCCN(C)CC3)cc2N1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.41
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
PARP1 P09874 3/20 0.38
LNPEP Q9UIQ6 1/20 0.36
DRD2 P14416 2/20 0.35
ADRA1D P25100 2/20 0.35
SLC6A4 P31645 2/20 0.35
ADRA1A P35348 2/20 0.35
ADRA1B P35368 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP2D6 P10635 1/20 0.35
HTR6 P50406 1/20 0.35
PRMT5 O14744 2/20 0.34
WDR77 Q9BQA1 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2566679 0.74 ACACB (0.46) HRH3PARP1CYP2D6PRMT5WDR77
SCHEMBL15881982 0.71 HRH3 (0.52) HRH3MAOAMAOBPARP1DRD2
SCHEMBL15880539 0.69 HRH3 (0.47) HRH3MAOAMAOBPARP1SMN1; SMN2
SCHEMBL15880537 0.69 HRH3 (0.47) HRH3MAOAMAOBPARP1SMN1; SMN2
SCHEMBL17311546 0.69 HRH3 (0.47) HRH3MAOAMAOBPARP1SMN1; SMN2
SCHEMBL5466386 0.67 FPR2 (0.51) HRH3MAOAMAOBSLC6A4SMN1; SMN2
SCHEMBL10686530 0.66 MAOA (0.46) HRH3MAOAMAOBPARP1SMN1; SMN2
SCHEMBL2561454 0.66 HRH3 (0.46) HRH3PARP1DRD2CYP2D6PRMT5
SCHEMBL13849617 0.65 HRH3 (0.54) HRH3SMN1; SMN2
SCHEMBL2560796 0.65 DRD2 (0.50) HRH3MAOAMAOBDRD2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960387-B1 ISOQUINOLINE ET BENZO[H]ISOQUINOLINE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF AS ANTAGONISTS OF HISTAMINE H3 RECEPTOR SANOFI SA (FR) 2011-11-02 EP claimed