SCHEMBL2561692

SCHEMBL2561692

CCCCn1nc(-c2ccccc2)c(OC(=O)OC)c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.44
MEN1 O00255 5/20 0.44
CYP1A2 P05177 2/20 0.44
MAPT P10636 1/20 0.44
NR1H3 Q13133 1/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TSHR P16473 2/20 0.41
CYP2C9 P11712 1/20 0.41
CRHBP P24387 1/20 0.41
CYP2C19 P33261 1/20 0.41
CRHR2 Q13324 1/20 0.41
SMPD1 P17405 1/20 0.41
HSF1 Q00613 1/20 0.41
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16500067 0.81 TP53 (0.48) KMT2AMEN1CYP1A2MAPTKDM4E
SCHEMBL12264902 0.81 KMT2A (0.50) KMT2AMEN1CYP1A2MAPTNR1H3
SCHEMBL14482152 0.77 MEN1 (0.56) KMT2AMEN1CYP1A2MAPTNR1H3
SCHEMBL2553897 0.76 MEN1 (0.58) KMT2AMEN1CYP1A2MAPTALDH1A1
SCHEMBL2560670 0.76 KMT2A (0.43) KMT2AMEN1MAPTKDM4EALDH1A1
SCHEMBL23403222 0.75 MEN1 (0.53) KMT2AMEN1CYP1A2MAPTNR1H3
SCHEMBL2560863 0.71 ALDH1A1 (0.55) KMT2AMEN1KDM4EALDH1A1HPGD
SCHEMBL2555919 0.71 SMN1; SMN2 (0.41) KMT2AMEN1MAPTALDH1A1LMNA
SCHEMBL23401883 0.70 MEN1 (0.53) KMT2AMEN1CYP1A2MAPTNR1H3
SCHEMBL2554340 0.69 KMT2A (0.56) KMT2AMEN1MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-B1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms Universität Münster (DE) 2015-02-25 EP disclosed
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed