SCHEMBL2553897

SCHEMBL2553897

COC(=O)Oc1c(-c2ccccc2)nn(-c2ccccc2)c1C

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
ALDH1A1 P00352 7/20 0.54
TSHR P16473 1/20 0.45
MAPT P10636 6/20 0.45
RAB9A P51151 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
NPC1 O15118 2/20 0.44
RXFP1 Q9HBX9 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 3/20 0.42
HPGD P15428 1/20 0.42
PDE4D Q08499 1/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2C19 P33261 3/20 0.42
CYP3A4 P08684 2/20 0.42
CYP1A2 P05177 1/20 0.42
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2560863 0.91 ALDH1A1 (0.55) MEN1KMT2AALDH1A1NPSR1SMN1; SMN2
SCHEMBL2557760 0.90 MEN1 (0.48) MEN1KMT2AALDH1A1MAPTRAB9A
SCHEMBL2557580 0.90 KMT2A (0.48) MEN1KMT2AALDH1A1TSHRMAPT
SCHEMBL16500135 0.87 ALDH1A1 (0.51) MEN1KMT2AALDH1A1MAPTRAB9A
SCHEMBL2554340 0.87 KMT2A (0.56) MEN1KMT2AALDH1A1TSHRMAPT
SCHEMBL16500067 0.83 TP53 (0.48) MEN1KMT2AALDH1A1MAPTNPSR1
SCHEMBL2561201 0.83 MEN1 (0.42) MEN1KMT2AALDH1A1TSHRMAPT
SCHEMBL2557260 0.83 KDM4E (0.48) MEN1KMT2AALDH1A1TSHRMAPT
SCHEMBL2560670 0.81 KMT2A (0.43) MEN1KMT2AALDH1A1TSHRMAPT
SCHEMBL2576433 0.80 TSHR (0.47) MEN1KMT2AALDH1A1TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-B1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms Universität Münster (DE) 2015-02-25 EP disclosed
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed