SCHEMBL25625908

SCHEMBL25625908

CSC1c2ccccc2OCC1NC(=O)Cc1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.48
GRM7 Q14831 1/20 0.46
LMNA P02545 1/20 0.45
XIAP P98170 1/20 0.43
TP53 P04637 1/20 0.43
PSMB5 P28074 2/20 0.42
HCRTR2 O43614 1/20 0.42
POLB P06746 1/20 0.42
AIMP2 Q13155 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAOB P27338 1/20 0.39
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182997 0.80 GRM7 (0.57) P2RX7GRM7XIAPHCRTR2
SCHEMBL21542223 0.80 GRM7 (0.57) P2RX7GRM7XIAPHCRTR2
SCHEMBL21542222 0.80 GRM7 (0.57) P2RX7GRM7XIAPHCRTR2
SCHEMBL20182824 0.75 LTB4R (0.56) GRM7PSMB5POLBAIMP2CYP1A2
SCHEMBL20182869 0.74 AIMP2 (0.56) GRM7PSMB5POLBAIMP2CYP1A2
SCHEMBL20182939 0.74 PSMB5 (0.50) P2RX7PSMB5POLBAIMP2CYP1A2
SCHEMBL20182774 0.73 PSMB5 (0.52) P2RX7PSMB5POLBAIMP2CYP1A2
SCHEMBL25626161 0.73 PSMB5 (0.49) P2RX7LMNAPSMB5POLBAIMP2
SCHEMBL20182785 0.73 AIMP2 (0.52) P2RX7GRM7PSMB5POLBAIMP2
SCHEMBL21542206 0.72 GRM7 (0.61) P2RX7GRM7POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3541812-B1 MGLUR7 AGONIST COMPOUNDS FOR TREATING MGLUR7- REGULATED DISEASES, DISORDERS, OR CONDITIONS TAKEDA PHARMACEUTICALS CO (JP) 2023-06-14 EP disclosed