SCHEMBL2564355

SCHEMBL2564355

NC1=NS(=O)(=O)c2cccc(Cl)c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.43
GRK5 P34947 1/20 0.43
TYRO3 Q06418 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
CXCR2 P25025 2/20 0.37
PNMT P11086 1/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
NOS3 P29474 2/20 0.33
GAA P10253 1/20 0.33
CXCR1 P25024 1/20 0.33
LMNA P02545 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
RECQL P46063 1/20 0.32
IDO1 P14902 1/20 0.32
NR4A2 P43354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4149675 0.81 RET (0.46) RETGRK5TYRO3DYRK1BCXCR2
SCHEMBL10996068 0.79 LMNA (0.41) CA12CA1CA2CA9CA4
SCHEMBL11090288 0.78 BACE1 (0.36) CXCR2CA12CA1CA2CA9
SCHEMBL8285729 0.78 RET (0.43) RETGRK5TYRO3DYRK1BCXCR2
SCHEMBL11165904 0.78 CXCR2 (0.37) CXCR2CA12CA1CA2CA9
SCHEMBL2573400 0.74 HSD17B10 (0.48) CXCR2CA1CA2CA9CA7
SCHEMBL13903578 0.74 RET (0.40) RETGRK5TYRO3DYRK1BCXCR2
SCHEMBL13903591 0.71 RET (0.38) RETGRK5TYRO3DYRK1BCXCR2
SCHEMBL13903622 0.71 RET (0.38) RETGRK5TYRO3DYRK1BCXCR2
SCHEMBL13903579 0.70 HTT (0.43) RETGRK5TYRO3DYRK1BCXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033984-B1 NEW SULPHONYL COMPOUNDS, METHOD OF PREPARING THE NEW COMPOUNDS, AS WELL AS APHICIDAL COMPOSITIONS ON THE BASIS OF THE NEW COMPOUNDS DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1984-06-06 EP claimed
US-4379157-A Sulphonyl compounds, method of preparing the new compounds, as well as aphicidal compositions on the basis of the new compounds DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1983-04-05 US claimed
JP-2006496-A None JP disclosed
EP-2148567-B1 A METHOD OF PROTECTING A PLANT PROPAGATION MATERIAL, A PLANT, AND/OR PLANT ORGANS SYNGENTA PARTICIPATIONS AG (CH) 2011-11-02 EP disclosed
US-20100173959-A1 METHOD OF PROTECTING A PLANT PROPAGATION MATERIAL, A PLANT, AND/OR PLANT ORGANS SYNGENTA CROP PROTECTION, INC. (US) 2010-07-08 US disclosed
WO-2009141065-A2 (1,2-BENZISOTHIAZOL-3-YL)(THIO)CARBAMATES AND (1,2-BENZISOTHIAZOL-3-YL)(THIO)OXAMATES AND THE OXIDATION FORMS THEREOF FOR USE AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2009-11-26 WO disclosed
JP-H026496-A ORGANIC PHOSPHORIC ACID AMIDE COMPOUND, ITS PRODUCTION AND HARMFUL ANIMAL-CONTROLLING AGENT CONTAINING THE SAME COMPOUND ISHIHARA SANGYO KAISHA LTD 1990-01-10 JP disclosed
US-4760076-A Inhibiting allergen-induced degranulation of peripheral leukocytes CIBA-GEIGY CORPORATION (US) 1988-07-26 US disclosed
US-4492705-A INSECTICIDE, MITICIDE CIBA-GEIGY CORPORATION (US) 1985-01-08 US disclosed
EP-0033984-B1 NEW SULPHONYL COMPOUNDS, METHOD OF PREPARING THE NEW COMPOUNDS, AS WELL AS APHICIDAL COMPOSITIONS ON THE BASIS OF THE NEW COMPOUNDS DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1984-06-06 EP disclosed
US-4379157-A Sulphonyl compounds, method of preparing the new compounds, as well as aphicidal compositions on the basis of the new compounds DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1983-04-05 US disclosed
EP-0033984-A1 New sulphonyl compounds, method of preparing the new compounds, as well as aphicidal compositions on the basis of the new compounds DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1981-08-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100173959-A1 METHOD OF PROTECTING A PLANT PROPAGATION MATERIAL, A PLANT, AND/OR PLANT ORGANS RER1, H1-0, H1-2 RET 3450/4885GRK5 2770/4885TYRO3 4716/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.