SCHEMBL2564655

SCHEMBL2564655

COC(=O)Oc1c(C(C)C)nn(-c2ccc(F)cc2)c1C

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.46
P2RX7 Q99572 3/20 0.43
PTGS2 P35354 2/20 0.40
SLC34A1 Q06495 1/20 0.39
NR3C1 P04150 2/20 0.38
ALDH1A1 P00352 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
POLB P06746 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ABHD16A O95870 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
CFTR P13569 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2559798 0.85 SLC34A1 (0.49) P2RX7PTGS2SLC34A1NR3C1ALDH1A1
SCHEMBL2561878 0.81 PDE4D (0.41) P2RX7PTGS2SLC34A1ALDH1A1L3MBTL1
SCHEMBL2554143 0.81 SLC34A1 (0.43) P2RX7PTGS2SLC34A1NR3C1LMNA
SCHEMBL12264385 0.81 PPARA (0.47) PPARAP2RX7PTGS2SLC34A1ALDH1A1
SCHEMBL2560863 0.79 ALDH1A1 (0.55) SLC34A1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL14482134 0.76 PPARA (0.56) PPARAP2RX7PTGS2ALDH1A1POLB
SCHEMBL28497651 0.75 CFTR (0.45) PPARAP2RX7MEN1KMT2ACFTR
SCHEMBL16500084 0.69 TSHR (0.43) P2RX7PTGS2ALDH1A1POLBMEN1
SCHEMBL12265091 0.69 PDE4D (0.58) PTGS2SLC34A1ALDH1A1L3MBTL1KDM4E
SCHEMBL2553897 0.68 MEN1 (0.58) ALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552895-B1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms Universität Münster (DE) 2015-02-25 EP disclosed
EP-2552895-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES Westfälische Wilhelms-Universität Münster (DE) 2013-02-06 EP disclosed
WO-2011120861-A1 PYRAZOLE SYNTHESIS BY COUPLING OF CARBOXYLIC ACID DERIVATIVES AND ENAMINES WESTFÄLISHE WILHELMS-UNIVERSITÄT MÜNSTER (DE) 2011-10-06 WO disclosed