SCHEMBL2566906

SCHEMBL2566906

CCNS(=O)(=O)c1ccc(F)cc1F

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.49
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
CXCR4 P61073 1/20 0.46
KAT6A Q92794 1/20 0.44
KMT2A Q03164 1/20 0.44
KCNH2 Q12809 1/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
MEP1B Q16820 1/20 0.43
USP2 O75604 1/20 0.43
ALOX5AP P20292 1/20 0.43
FEN1 P39748 1/20 0.43
GLA P06280 1/20 0.43
BRD4 O60885 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26073802 0.81 MAPT (0.49) CCR2ALDH1A1LMNAPOLBCXCR4
SCHEMBL1013641 0.80 SMN1; SMN2 (0.43) ALDH1A1KMT2ASMN1; SMN2MEP1BUSP2
SCHEMBL2371266 0.79 CCR2 (0.53) CCR2ALDH1A1LMNAPOLBKAT6A
SCHEMBL1775171 0.79 LMNA (0.51) CCR2ALDH1A1LMNAPOLBCXCR4
SCHEMBL22233802 0.78 KMT2A (0.55) CCR2ALDH1A1LMNAPOLBCXCR4
SCHEMBL14011214 0.78 GBA1 (0.55) ALDH1A1KAT6AKMT2AALOX5APFEN1
SCHEMBL776801 0.77 AKR1B1 (0.44) CCR2ALDH1A1POLBKAT6AKCNH2
SCHEMBL24429412 0.76 CCR2 (0.50) CCR2ALDH1A1LMNAPOLBCXCR4
SCHEMBL2941883 0.76 LMNA (0.52) ALDH1A1LMNACXCR4KMT2AKCNH2
SCHEMBL7010992 0.76 MEN1 (0.53) ALDH1A1LMNAPOLBCXCR4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11976075-B2 Inhibitors of the MYST family of lysine acetyl transferases Isosterix, Inc. 2024-05-07 US disclosed
WO-2023192817-A1 INHIBITORS OF THE MYST FAMILY OF LYSINE ACETYL TRANSFERASES Isosterix, Inc. (US) 2023-10-05 WO disclosed
US-20230303580-A1 INHIBITORS OF THE MYST FAMILY OF LYSINE ACETYL TRANSFERASES Isosterix, Inc. 2023-09-28 US disclosed
EP-2556069-A1 PYRIMIDINYLPIPERIDINYLOXYPYRIDINONE ANALOGUES AS GPR119 MODULATORS Bristol-Myers Squibb Company (US) 2013-02-13 EP disclosed
WO-2011127106-A1 PYRIMIDINYLPIPERIDINYLOXYPYRIDINONE ANALOGUES AS GPR119 MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-10-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303580-A1 INHIBITORS OF THE MYST FAMILY OF LYSINE ACETYL TRANSFERASES KAT6A, KAT6B, KAT2A CCR2 4769/4885ALDH1A1 1618/4885LMNA 2088/4885
US-11976075-B2 Inhibitors of the MYST family of lysine acetyl transferases KAT6A, KAT6B, KAT2A CCR2 4769/4885ALDH1A1 1618/4885LMNA 2088/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.